SCHEMBL28889290

SCHEMBL28889290

O=C(NC(=S)NC1CC1)C(c1cccc(F)c1)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
PHGDH O43175 2/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CRHR1 P34998 1/20 0.37
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37
BRD4 O60885 1/20 0.37
IDH1 O75874 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4D Q08499 1/20 0.36
UBE2M P61081 1/20 0.36
DCUN1D1 Q96GG9 1/20 0.36
GALR3 O60755 1/20 0.36
SMYD3 Q9H7B4 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
OPRL1 P41146 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889357 0.88 ALDH1A1 (0.39) LMNAPHGDHALDH1A1GRIN1GRIN2B
SCHEMBL29941818 0.87 HDAC4 (0.41) LMNAPHGDHHDAC4HDAC7HDAC5
SCHEMBL28889342 0.85 OPRM1 (0.40) LMNAPHGDHHDAC4HDAC7HDAC5
SCHEMBL28889315 0.85 PHGDH (0.39) LMNAPHGDHALDH1A1CRHR1
SCHEMBL28889259 0.85 HDAC4 (0.42) HDAC4HDAC7HDAC5KMT2ANPSR1
SCHEMBL28889177 0.83 HDAC4 (0.40) LMNAPHGDHHDAC4HDAC7HDAC5
SCHEMBL29893652 0.83 PDE4B (0.38) LMNAPHGDHALDH1A1CRHR1PDE4B
SCHEMBL28889234 0.83 PDE4B (0.38) LMNAPHGDHALDH1A1CRHR1PDE4B
SCHEMBL28889330 0.83 ALDH1A1 (0.44) LMNAPHGDHALDH1A1CRHR1IDH1
SCHEMBL28889214 0.82 HDAC4 (0.39) PHGDHHDAC4HDAC7HDAC5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed