SCHEMBL28896573

SCHEMBL28896573

CCOC(=O)c1[nH]ccc1NCC(CN)OCC(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33
KMT2A Q03164 1/20 0.33
NUDT1 P36639 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PDK1 Q15118 1/20 0.32
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32
LMNA P02545 3/20 0.32
POLB P06746 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28896256 0.84 MAPT (0.36) KDM4ENPSR1SMN1; SMN2PDK1PDK2
SCHEMBL28896575 0.84 LMNA (0.33) KDM4EKMT2ANUDT1SMN1; SMN2ALDH1A1
SCHEMBL28896488 0.80 SMN1; SMN2 (0.36) KDM4ENPSR1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL28896261 0.79 KDM4E (0.34) KDM4ENPSR1JAK2JAK3KMT2A
SCHEMBL28896250 0.77 PTGER4 (0.38) KDM4ENPSR1JAK2JAK3KMT2A
SCHEMBL1536614 0.76 ALDH1A1 (0.44) KDM4EKMT2ANUDT1SMN1; SMN2ALDH1A1
SCHEMBL28896207 0.76 KMT2A (0.34) KDM4ENPSR1KMT2ANUDT1SMN1; SMN2
SCHEMBL28896275 0.73 KDM4E (0.35) KDM4ENPSR1KMT2ANUDT1SMN1; SMN2
SCHEMBL29211269 0.72 KMT2A (0.34) KDM4ENPSR1KMT2ANUDT1SMN1; SMN2
SCHEMBL4200796 0.71 ALDH1A1 (0.45) KDM4EKMT2ANUDT1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403584-B 2-thio-2, 3-dihydropyrimidine-4-one derivatives, pharmaceutical compositions, preparation methods and applications thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115403584-A 2-thio-2, 3-dihydropyrimidine-4-one derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-29 CN disclosed