SCHEMBL28899709

SCHEMBL28899709

O=C(O)c1cc2cccc([N+](=O)[O-])c2n1N1CCOCC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.50
APEX1 P27695 1/20 0.42
KDM4E B2RXH2 3/20 0.41
MAPT P10636 4/20 0.40
PKM P14618 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
MCL1 Q07820 1/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 1/20 0.39
POLB P06746 1/20 0.39
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CASP6 P55212 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28461691 0.84 MAPT (0.43) CCR2KDM4EMAPTKMT2AMEN1
SCHEMBL28899797 0.77 FBP1 (0.51) KMT2A
SCHEMBL28294933 0.74 CCR2 (0.55) CCR2APEX1CYP1A2MCL1KMT2A
SCHEMBL3255649 0.74 CCR2 (0.55) CCR2APEX1KDM4EMCL1ALDH1A1
SCHEMBL27964872 0.74 CCR2 (0.58) CCR2APEX1MCL1KMT2AMEN1
SCHEMBL7993476 0.71 CCR2 (0.64) CCR2APEX1MAPTCYP1A2MCL1
SCHEMBL28079176 0.68 CCR2 (0.54) CCR2APEX1MAPTMCL1ALDH1A1
SCHEMBL16653775 0.67 KDM4E (0.57) KDM4EMAPTPKMCYP1A2CYP2C9
SCHEMBL5266320 0.65 CCR2 (0.46) CCR2APEX1KDM4EMAPTKMT2A
SCHEMBL6141958 0.65 HRH4 (0.43) MAPTPKMCYP1A2CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098846-B N-acyl sulfonamide FBPase inhibitor, preparation method thereof, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-10-09 CN disclosed