SCHEMBL28906211

SCHEMBL28906211

Cn1nnc(-c2ncc(C(F)(F)F)cn2)c1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 1/20 0.41
AKR1C3 P42330 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
AGBL2 Q5U5Z8 1/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
KDM2B Q8NHM5 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
HDAC4 P56524 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
HCAR3 P49019 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28906191 0.85 LMNA (0.41) IKBKEAKR1C3L3MBTL1KMT2AMEN1
SCHEMBL26097267 0.75 CYP1A2 (0.35) IKBKEAGBL2ALDH1A1KDM4ELMNA
SCHEMBL24867893 0.73 MAPK14 (0.38)
SCHEMBL28906199 0.70 LMNA (0.38) AKR1C3KMT2AMEN1ALDH1A1LMNA
Trifluoroacetic Acid SCHEMBL30455778 0.69 LDHA (0.34) IKBKEAKR1C3KMT2AMEN1GPBAR1
SCHEMBL16708689 0.67 POLB (0.45) KMT2AMEN1HPGDSMN1; SMN2ALDH1A1
SCHEMBL23363075 0.67 L3MBTL1 (0.38) L3MBTL1KMT2AMEN1GPBAR1SMN1; SMN2
SCHEMBL25224521 0.66 LDHA (0.35) KMT2AMEN1HDAC4POLBHCAR3
SCHEMBL23363199 0.66 ALDH1A1 (0.42) KMT2AMEN1ALDH1A1KDM4EKDM2B
SCHEMBL21590723 0.66 NPC1 (0.45) KMT2AMEN1AGBL2GPBAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461337-A Novel triazolyl derivatives as GABA A alpha 5 PAM 豪夫迈·罗氏有限公司 2022-12-09 CN disclosed