SCHEMBL28906365

SCHEMBL28906365

FC(F)(F)c1ccc(-c2[nH]c3ccccc3c2Cc2c(-c3ccc(C(F)(F)F)cc3)[nH]c3ccccc23)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.50
HTR2C P28335 4/20 0.50
KIF11 P52732 3/20 0.50
DRD2 P14416 3/20 0.50
MGAM O43451 1/20 0.45
GAA P10253 1/20 0.45
SI P14410 1/20 0.45
MGAM2 Q2M2H8 1/20 0.45
MCL1 Q07820 1/20 0.44
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44
TUBA4A P68366 1/20 0.44
TUBB4B P68371 1/20 0.44
TUBB3 Q13509 1/20 0.44
TUBB2A Q13885 1/20 0.44
TUBB8 Q3ZCM7 1/20 0.44
TUBA3E Q6PEY2 1/20 0.44
TUBA1A Q71U36 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28906353 0.81 HTR2A (0.61) HTR2AHTR2CDRD2TUBB4ATUBB
SCHEMBL28906516 0.81 HTR2A (0.62) HTR2AHTR2CDRD2TUBB4ATUBB
SCHEMBL27549075 0.79 KIF11 (0.51) KIF11MGAMGAASIMGAM2
SCHEMBL5635637 0.78 KIF11 (0.47) KIF11MGAMGAASIMGAM2
SCHEMBL28906369 0.78 MAPT (0.55) HTR2AHTR2CDRD2TUBB4ATUBB
SCHEMBL28906371 0.78 HTR2A (0.61) HTR2AHTR2CDRD2TUBB4ATUBB
SCHEMBL28906377 0.78 PTGS2 (0.49) HTR2AHTR2CDRD2TUBB4ATUBB
SCHEMBL28906514 0.74 KDM4E (0.58) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL10443772 0.74 TUBB4A (0.64) HTR2AHTR2CKIF11DRD2TUBB4A
SCHEMBL607944 0.72 KIF11 (0.75) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304533-B Bisindolemethane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2024-04-12 CN disclosed
CN-117567447-A Thiophene-containing bis-indolomethane type a-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2024-02-20 CN disclosed
CN-115304533-A Bis-indole methane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2022-11-08 CN disclosed