SCHEMBL28906480

SCHEMBL28906480

CCc1cc(C(=O)OC)c(F)c(Cl)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 3/20 0.40
KDM4E B2RXH2 2/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 2/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
ABL1 P00519 1/20 0.37
ALDH1A1 P00352 2/20 0.36
NQO2 P16083 5/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28906546 0.82 KEAP1 (0.47) KDM4ERAB9ASMN1; SMN2ALDH1A1
SCHEMBL21349700 0.82 KDM4E (0.53) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL21349339 0.81 KDM4E (0.47) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL21348932 0.79 ALDH1A1 (0.50) KDM4ESMN1; SMN2L3MBTL1ABL1ALDH1A1
SCHEMBL31320124 0.79 ALDH1A1 (0.50) KDM4ESMN1; SMN2L3MBTL1ABL1ALDH1A1
SCHEMBL12590479 0.76 MAPT (0.44) PLA2G2AKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL28906484 0.75 MAPT (0.42) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL21551592 0.75 PLA2G2A (0.43) PLA2G2AKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL30931812 0.75 PLA2G2A (0.43) PLA2G2AKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL28906556 0.73 JMJD6 (0.42) PLA2G2AKDM4EMAPTL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304623-A Pyrimido-cyclic derivative and application thereof in medicine 四川海思科制药有限公司 2022-11-08 CN disclosed