SCHEMBL28906705

SCHEMBL28906705

O=CN1CCN(c2cccc(Oc3ccccc3)c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP14 Q460N5 2/20 0.48
PARP10 Q53GL7 2/20 0.48
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
SLC6A3 Q01959 1/20 0.47
MAPT P10636 4/20 0.46
CRHBP P24387 1/20 0.46
HTT P42858 1/20 0.46
CRHR2 Q13324 1/20 0.46
LTA4H P09960 1/20 0.45
MAOB P27338 1/20 0.44
LMNA P02545 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
FFAR1 O14842 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28522648 0.87 LTA4H (0.60) PARP14PARP10MAPTCRHBPHTT
SCHEMBL2359935 0.84 ADRB1 (0.59) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL29786218 0.84 ADRB1 (0.59) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL11510734 0.81 SLC6A2 (0.52) PARP14PARP10SLC6A2SLC6A4SLC6A3
SCHEMBL4052281 0.80 AKR1C3 (0.52) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL30228382 0.80 SLC6A2 (0.51) PARP14PARP10SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL27859960 0.79 CYP2C9 (0.50) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL20708552 0.78 ALDH1A1 (0.60) SLC6A4MAPTHTTLMNAALDH1A1
SCHEMBL23222244 0.77 DRD2 (0.56) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL4671113 0.77 SLC6A2 (0.49) PARP14PARP10SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112341396-B Novel monoacylglycerol esterase inhibitor and preparation method and application thereof 四川大学华西医院 2022-07-26 CN disclosed
CN-112341396-A Novel monoacylglycerol esterase inhibitor and preparation method and application thereof 四川大学华西医院 2021-02-09 CN disclosed