SCHEMBL2892908

SCHEMBL2892908

Cc1c(C(=O)O)sc2c(F)cc(F)cc12

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 10/20 0.46
PKM P14618 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
BCKDK O14874 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.34
MKNK2 Q9HBH9 2/20 0.34
MKNK1 Q9BUB5 1/20 0.34
AKR1B1 P15121 1/20 0.34
KDM4E B2RXH2 1/20 0.33
PTGER4 P35408 1/20 0.33
BCL2L1 Q07817 1/20 0.33
MCL1 Q07820 1/20 0.33
TBXAS1 P24557 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31126960 0.80 ALDH1A1 (0.45) NPSR1TRPM8KDM4E
SCHEMBL2889379 0.77 GPR35 (0.44) GPR35PKMNPSR1RXFP1MCL1
SCHEMBL2893771 0.73 GPR35 (0.58) GPR35PKMNPSR1RXFP1BCKDK
SCHEMBL31126901 0.71 ERN1 (0.34)
SCHEMBL31126894 0.71 DHODH (0.32) AKR1B1
SCHEMBL20561760 0.71 GPR35 (0.42) GPR35PKMNPSR1RXFP1BCKDK
SCHEMBL2895162 0.70 BCKDK (0.67) GPR35PKMNPSR1RXFP1BCKDK
SCHEMBL3687153 0.68 GPR35 (0.59) GPR35PKMNPSR1RXFP1BCKDK
SCHEMBL31207537 0.67 GPR35 (0.48) GPR35PKMNPSR1RXFP1MKNK2
SCHEMBL2610279 0.67 GPR35 (0.51) GPR35PKMNPSR1RXFP1BCKDK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732477-B2 N-(1-azabicyclo[2.2.2]oct-3-yl)-heteroaryl carboxamides; alpha 7-nicotinic acetylcholine receptors (nAChR) agonists; improving perception, concentration, learning and memory; neuropathic pain; acute and chronic pain BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-06-08 US disclosed