SCHEMBL28958322

SCHEMBL28958322

O=C1SCCN1Cc1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 1/20 0.50
CHRNA1 P02708 1/20 0.43
CHRNA7 P36544 1/20 0.43
NPC1 O15118 1/20 0.43
HTT P42858 1/20 0.43
MAPK1 P28482 1/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HSD11B1 P28845 1/20 0.41
POLB P06746 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9514131 0.86 ALDH1A1 (0.60) ALDH1A1KDM4ECHRNA1CHRNA7NPC1
SCHEMBL9511632 0.83 HTT (0.59) ALDH1A1KDM4EHTTPOLBKMT2A
SCHEMBL4182979 0.82 MAPK1 (0.57) ALDH1A1KDM4EMAPK1POLBKMT2A
SCHEMBL9512641 0.79 POLB (0.62) ALDH1A1MAPK1POLBGRM2KMT2A
SCHEMBL9741850 0.79 ALDH1A1 (0.49) ALDH1A1KDM4ECHRNA1CHRNA7NPC1
SCHEMBL28958218 0.79 POLB (0.56) ALDH1A1CHRNA1CHRNA7NPC1HTT
SCHEMBL9743824 0.79 ALDH1A1 (0.44) ALDH1A1CHRNA1CHRNA7NPC1HTT
SCHEMBL9511103 0.78 KDM4E (0.57) ALDH1A1KDM4EHDAC1HDAC6POLB
SCHEMBL14094206 0.75 ALDH1A1 (0.41) ALDH1A1KDM4ECHRNA1CHRNA7NPC1
SCHEMBL9413138 0.74 MAPT (0.56) ALDH1A1KDM4ENPC1HTTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110294719-B Synthesis method of thiazolidone compound 五邑大学 2023-02-28 CN disclosed
CN-114409680-A PPAR agonist and application thereof 上海怡立舍生物技术有限公司 2022-04-29 CN disclosed
CN-108250058-B PPAR agonists and their use in the treatment of Alzheimer's disease and other diseases 上海怡立舍生物技术有限公司 2022-02-11 CN disclosed