SCHEMBL9741850

SCHEMBL9741850

O=C1SCCN1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.49
P2RX3 P56373 1/20 0.46
HDAC1 Q13547 1/20 0.44
NPC1 O15118 1/20 0.43
OPRL1 P41146 1/20 0.41
CHRNA1 P02708 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRM5 P08912 1/20 0.40
HIF1A Q16665 1/20 0.40
EPAS1 Q99814 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HTT P42858 1/20 0.40
COMT P21964 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
CHKA P35790 1/20 0.40
EP300 Q09472 1/20 0.39
CREBBP Q92793 1/20 0.39
KAT2A Q92830 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28958218 0.84 POLB (0.56) ALDH1A1HDAC1NPC1CHRNA1CHRNA7
SCHEMBL9742340 0.82 KDM4E (0.54) ALDH1A1KDM4E
SCHEMBL9514131 0.82 ALDH1A1 (0.60) ALDH1A1KDM4ENPC1CHRNA1CHRNA7
SCHEMBL28958322 0.79 ALDH1A1 (0.50) ALDH1A1KDM4EHDAC1NPC1CHRNA1
SCHEMBL9511632 0.79 HTT (0.59) ALDH1A1KDM4EHTTPOLB
SCHEMBL4182979 0.78 MAPK1 (0.57) ALDH1A1KDM4EL3MBTL1POLB
SCHEMBL9743824 0.75 ALDH1A1 (0.44) ALDH1A1NPC1CHRNA1CHRNA7HIF1A
SCHEMBL9511103 0.74 KDM4E (0.57) ALDH1A1KDM4EHDAC1POLB
SCHEMBL23310507 0.73 L3MBTL1 (0.59) ALDH1A1KDM4EHDAC1L3MBTL1CHKA
SCHEMBL9742351 0.73 KMT2A (0.50) ALDH1A1KDM4ECOMTSIRT2SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5169859-A Antisecretory or antiulcer agents RICHTER GEDEON VEGYESZETI GYAR RT (HU) 1992-12-08 US disclosed
EP-0455774-A1 THIAZOLIDINONE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME RICHTER GEDEON VEGYESZETI GYAR R.T. (HU) 1991-11-13 EP disclosed
WO-1991008203-A1 NOVEL THIAZOLIDINONE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME Richter Gedeon Vegyészeti Gyár Rt. (HU) 1991-06-13 WO disclosed