SCHEMBL29009207

SCHEMBL29009207

COc1ccc(NC(=O)C2CC(c3ccccc3)NC2=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.57
MAPT P10636 1/20 0.54
GRIN2B Q13224 1/20 0.48
MAP2K1 Q02750 2/20 0.48
RAB9A P51151 3/20 0.46
NPC1 O15118 2/20 0.46
ACHE P22303 1/20 0.46
BACE1 P56817 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 1/20 0.45
CYP2C19 P33261 2/20 0.45
TP53 P04637 1/20 0.45
CYP2C9 P11712 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30466244 0.94 MAP2K1 (0.51) USP2MAPTMAP2K1RAB9ANPC1
SCHEMBL29009181 0.88 FPR2 (0.53) USP2MAPTMAP2K1MEN1KMT2A
SCHEMBL29009179 0.78 MMP1 (0.50) MAPTBACE1MEN1KMT2ACYP2C19
SCHEMBL29009153 0.78 CYP2D6 (0.44) MEN1KMT2APOLBLMNA
SCHEMBL10123277 0.75 DEGS1 (0.70) USP2MAPTGRIN2BRAB9ANPC1
SCHEMBL871979 0.75 DEGS1 (0.70) USP2MAPTGRIN2BRAB9ANPC1
SCHEMBL4242864 0.72 NPC1 (0.50) USP2MAPTGRIN2BRAB9ANPC1
SCHEMBL29009157 0.71 RAB9A (0.55) USP2MAPTRAB9ANPC1MEN1
SCHEMBL7726470 0.69 MAPK1 (0.61) MAP2K1RAB9ANPC1POLB
SCHEMBL30466251 0.68 CHRNA7 (0.48) USP2MAPTMAP2K1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116217458-A 2-carbonyl-5-phenylpyrrole compound, preparation method, application and derivative thereof, and pharmaceutical composition 湖北民族大学 2023-06-06 CN disclosed