SCHEMBL29037153

SCHEMBL29037153

NC(=O)OCc1cc(F)ccc1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.42
PKM P14618 1/20 0.41
FFAR1 O14842 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
MMP2 P08253 2/20 0.39
MMP12 P39900 2/20 0.39
MMP1 P03956 1/20 0.39
MMP9 P14780 1/20 0.39
IDO1 P14902 2/20 0.36
AGXT P21549 2/20 0.36
NQO1 P15559 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PARP10 Q53GL7 2/20 0.35
POLB P06746 1/20 0.34
PIN1 Q13526 1/20 0.34
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14448981 0.83 ALDH1A1 (0.41) GRM5PKMFFAR1FFAR4MMP2
SCHEMBL30881188 0.83 ALDH1A1 (0.41) GRM5PKMFFAR1FFAR4MMP2
SCHEMBL28532155 0.80 NQO1 (0.36) PKMFFAR4MMP2MMP12MMP1
SCHEMBL5969470 0.80 GRM5 (0.42) GRM5MMP2MMP12MMP1MMP9
SCHEMBL23093403 0.80 MMP2 (0.39) PKMFFAR1FFAR4MMP2MMP12
SCHEMBL6629935 0.80 L3MBTL1 (0.44) PKMFFAR1FFAR4MMP2MMP12
SCHEMBL28954128 0.80 IDO1 (0.42) IDO1ALDH1A1NPSR1HSD17B10MAOB
SCHEMBL28717892 0.78 IDO1 (0.41) GRM5MMP2MMP12MMP1MMP9
SCHEMBL15524379 0.77 ICMT (0.43) PKMFFAR1FFAR4PIN1MPO
SCHEMBL114463 0.75 PARP10 (0.57) PKMFFAR1FFAR4MMP2MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111566103-B Aminoimidazopyrazines as kinase inhibitors 百时美施贵宝公司 2023-06-23 CN disclosed
CN-110520423-B Aminotriazolopyridines as kinase inhibitors 百时美施贵宝公司 2022-08-23 CN disclosed
CN-111566103-A Aminoimidazopyrazines as kinase inhibitors 百时美施贵宝公司 2020-08-21 CN disclosed