SCHEMBL30508200

SCHEMBL30508200

Nc1ncc(-c2ccc3nn(CCN4CCC(F)(F)CC4)cc3c2)cc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
IKBKE Q14164 1/20 0.39
TBK1 Q9UHD2 1/20 0.39
PIK3C3 Q8NEB9 1/20 0.39
MCHR1 Q99705 2/20 0.38
KDM5A P29375 2/20 0.37
KDM4C Q9H3R0 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
BMPR1B O00238 7/20 0.35
BMPR1A P36894 7/20 0.35
TGFBR1 P36897 7/20 0.35
ACVRL1 P37023 7/20 0.35
ACVR1 Q04771 7/20 0.35
PIK3CA P42336 2/20 0.35
MET P08581 1/20 0.35
S1PR1 P21453 1/20 0.35
AXL P30530 1/20 0.34
MERTK Q12866 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30508316 0.90 HDAC3 (0.41) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL29041963 0.90 HDAC3 (0.41) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508285 0.88 HDAC3 (0.55) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508332 0.87 BMPR1B (0.51) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL29042097 0.78 HDAC3 (0.52) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508338 0.78 HDAC3 (0.52) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508377 0.77 BMPR1B (0.61) HDAC3HDAC1HDAC2IKBKETBK1
SCHEMBL30508228 0.75 BMPR1B (0.43) PIK3C3BMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL29041989 0.71 MCHR1 (0.39) HDAC3HDAC1HDAC2MCHR1
SCHEMBL30508339 0.69 MET (0.44) PIK3C3BMPR1BBMPR1ATGFBR1ACVRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed