SCHEMBL29067977

SCHEMBL29067977

O=C(O)C[C@@H]1CNCC(F)(F)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 2/20 0.50
GABRA5 P31644 2/20 0.50
GABRB2 P47870 2/20 0.50
SLC6A12 P48065 2/20 0.50
SLC6A11 P48066 2/20 0.50
SLC6A13 Q9NSD5 2/20 0.50
GABRA1 P14867 1/20 0.50
GABRR1 P24046 1/20 0.50
GABRA4 P48169 1/20 0.50
ARG1 P05089 1/20 0.37
APLNR P35414 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
GRM2 Q14416 2/20 0.33
GRM5 P41594 1/20 0.33
GRM1 Q13255 1/20 0.33
SLC1A2 P43004 2/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29067981 1.00 SLC6A1 (0.50) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
Hydrochloric Acid SCHEMBL29180516 0.98 SLC6A12 (0.48) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
Hydrochloric Acid SCHEMBL29180517 0.98 SLC6A12 (0.48) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL29068028 0.83 ARG1 (0.43) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL29068055 0.83 ARG1 (0.43) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL15114485 0.79 APLNR (0.50) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL29067928 0.79 BRD4 (0.37) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL29067925 0.79 BRD4 (0.37) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL30452244 0.79 BRD4 (0.37) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL21111172 0.78 PTGIR (0.35) SLC6A1GABRA5GABRB2SLC6A12SLC6A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024022314-A1 TRIAZOLE COMPOUNDS AND USE THEREOF AS LPAR1 ANTAGONIST 武汉人福创新药物研发中心有限公司 2024-02-01 WO disclosed
CN-116669727-A Triazole-pyridinyl substituted azacyclohexylacetic acid compounds as LPA receptor antagonists 唯久生物有限公司 2023-08-29 CN disclosed