SCHEMBL29068134

SCHEMBL29068134

c1ccc(COc2ccc(-n3cccn3)cn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
NOTUM Q6P988 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
PKM P14618 1/20 0.40
ALKBH1 Q13686 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
LMNA P02545 1/20 0.39
FFAR1 O14842 1/20 0.38
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12989014 0.81 LMNA (0.50) DRD2DRD4DRD3NOTUMPKM
SCHEMBL20764923 0.81 NOTUM (0.45) NOTUMHRH3PKMKDM4EALDH1A1
SCHEMBL13723894 0.77 NOTUM (0.47) NOTUMHRH3KDM4EALDH1A1MAPK1
SCHEMBL15056311 0.74 KAT6A (0.45) DRD2DRD4DRD3NOTUMLMNA
SCHEMBL30500456 0.74 CHRNB2 (0.46) PKMKDM4EALDH1A1MAPK1FFAR1
SCHEMBL29068037 0.74 CHRNB2 (0.46) PKMKDM4EALDH1A1MAPK1FFAR1
SCHEMBL5759590 0.73 ALDH1A1 (0.47) KDM4EALDH1A1MAPK1LMNANPC1
SCHEMBL12989738 0.71 LMNA (0.50) ALKBH1LMNANPC1GLARAB9A
SCHEMBL28289846 0.71 PKM (0.40) PKMLMNAFFAR1GABRPGABRD
SCHEMBL31310179 0.71 NOTUM (0.46) NOTUMPKMLMNAFFAR1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116669727-A Triazole-pyridinyl substituted azacyclohexylacetic acid compounds as LPA receptor antagonists 唯久生物有限公司 2023-08-29 CN disclosed