SCHEMBL29072197

SCHEMBL29072197

COc1ccc(CNc2nc(Cc3ccc(OC)cc3)nc(N)c2N)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.50
ALDH1A1 P00352 1/20 0.48
CYP2D6 P10635 1/20 0.48
ATM Q13315 1/20 0.48
MAPT P10636 2/20 0.46
NCF1 P14598 1/20 0.46
MPO P05164 1/20 0.44
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
PRUNE1 Q86TP1 1/20 0.43
EGFR P00533 2/20 0.43
POLB P06746 1/20 0.43
NR2F2 P24468 1/20 0.43
HTR6 P50406 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25379641 0.82 MAPT (0.64) ALDH1A1MAPTEGFRNPSR1
SCHEMBL28391873 0.79 ALDH1A1 (0.54) ALDH1A1CYP2D6ATMMAPTMPO
SCHEMBL4864671 0.75 APP (0.70) APPALDH1A1CYP2D6MAPTNCF1
SCHEMBL28323063 0.75 ACP1 (0.44) APPNCF1HTR6
SCHEMBL3391705 0.74 APP (0.61) APPALDH1A1CYP2D6ATMNCF1
SCHEMBL23175129 0.73 LMNA (0.70) ALDH1A1CYP2D6ATMMAPTPOLB
SCHEMBL31410965 0.72 APP (0.60) APPMAPTNCF1
SCHEMBL34461806 0.71 ALDH1A1 (0.65) ALDH1A1CYP2D6ATMMAPTPOLB
SCHEMBL7172603 0.71 APP (0.51) APPMAPTNCF1PRUNE1EGFR
SCHEMBL3953843 0.71 APP (0.51) APPMAPTNCF1PRUNE1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116693458-A Cycloalkyl or heterocyclyl substituted heteroaryl compounds, compositions and uses thereof 深圳市塔吉瑞生物医药有限公司 2023-09-05 CN disclosed