SCHEMBL29073376

SCHEMBL29073376

NC(=O)OC1Cc2ncccc2N(c2ccc(C(F)(F)F)cc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.38
ROCK2 O75116 1/20 0.38
PDE4B Q07343 1/20 0.36
TRPV1 Q8NER1 6/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 2/20 0.35
TSHR P16473 1/20 0.35
TRPA1 O75762 1/20 0.35
AADAT Q8N5Z0 1/20 0.34
SLC6A7 Q99884 1/20 0.34
ELANE P08246 1/20 0.34
RPS6KB1 P23443 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.33
FPR1 P21462 1/20 0.33
FPR2 P25090 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29073342 0.83 TRPA1 (0.39) SLC6A2ROCK2PDE4BTRPV1ALDH1A1
SCHEMBL29073451 0.83 SLC6A2 (0.52) SLC6A2AADAT
SCHEMBL5362433 0.80 TBXAS1 (0.33) ALDH1A1AADAT
SCHEMBL29073370 0.79 SLC6A2 (0.38) SLC6A2AADATFPR1FPR2
SCHEMBL29073325 0.79 SLC6A2 (0.38) SLC6A2TRPV1AADATRPS6KB1TRPM8
SCHEMBL25331737 0.78 PDE4B (0.40) SLC6A2PDE4BTRPV1ALDH1A1HTT
SCHEMBL27057694 0.76 SLC6A2 (0.39) SLC6A2PDE4BTRPV1FPR1FPR2
SCHEMBL30767936 0.76 SLC6A2 (0.39) SLC6A2PDE4BTRPV1FPR1FPR2
SCHEMBL29073363 0.75 AADAT (0.41) SLC6A2AADAT
SCHEMBL31596872 0.73 ROCK2 (0.42) ROCK2PDE4BTRPV1TRPA1SLC6A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116783165-A 1,2,3, 4-tetrahydroquinoline derivatives as YAP/TAZ-TEAD activation inhibitors for the treatment of cancer 天主教鲁汶大学 2023-09-19 CN disclosed