SCHEMBL2908175

SCHEMBL2908175

CC(=O)CC(=O)Nc1cc(Br)c(NC(=O)CC(C)=O)cc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.47
ALDH1A1 P00352 5/20 0.46
KMT2A Q03164 5/20 0.46
MEN1 O00255 3/20 0.46
LMNA P02545 2/20 0.46
HTT P42858 2/20 0.46
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
RAB9A P51151 2/20 0.44
PAX8 Q06710 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
HIF1A Q16665 1/20 0.43
CA4 P22748 1/20 0.43
CA7 P43166 1/20 0.43
HPGD P15428 2/20 0.41
GAA P10253 1/20 0.41
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904641 0.82 KMT2A (0.55) MAPTALDH1A1KMT2AMEN1LMNA
SCHEMBL10386482 0.82 MAPT (0.41) MAPTALDH1A1KMT2AMEN1LMNA
SCHEMBL1116483 0.81 ALDH1A1 (0.52) MAPTALDH1A1KMT2AMEN1LMNA
SCHEMBL1116453 0.79 LMNA (0.58) MAPTALDH1A1KMT2AMEN1LMNA
SCHEMBL18750435 0.78 CA1 (0.56) MAPTALDH1A1LMNAHTTCA1
SCHEMBL2909396 0.77 MEN1 (0.55) MAPTALDH1A1KMT2AMEN1LMNA
SCHEMBL10386483 0.75 MAPT (0.35) MAPTALDH1A1KMT2AMEN1LMNA
SCHEMBL2914539 0.75 ALDH1A1 (0.54) MAPTALDH1A1KMT2AMEN1LMNA
SCHEMBL2911960 0.75 ALDH1A1 (0.50) MAPTALDH1A1KMT2AMEN1LMNA
SCHEMBL1128719 0.74 MAPT (0.60) MAPTALDH1A1KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6756486-B1 LAKED DISAZO YELLOW PIGMENTS HAVING DESIRABLE GREEN SHADE, HEAT STABILITY, GOOD STRENGTH, BLEED RESISTANCE, MIGRATION RESISTANCE, AND LOW OR NO TOXICITY ENGELHARD CORPORATION 2004-06-29 US claimed
EP-1668080-B1 NON-MIGRATING MEALLIZED DISAZO GREEN SHADE YELLOW PIGMENT ENGELHARD CORP (US) 2010-08-11 EP disclosed
EP-1668080-A1 NON-MIGRATING MEALLIZED DISAZO GREEN SHADE YELLOW PIGMENT Engelhard Corporation (US) 2006-06-14 EP disclosed
WO-2005033212-A1 NON-MIGRATING MEALLIZED DISAZO GREEN SHADE YELLOW PIGMENT ENGELHARD CORPORATION (US) 2005-04-14 WO disclosed
US-6756486-B1 LAKED DISAZO YELLOW PIGMENTS HAVING DESIRABLE GREEN SHADE, HEAT STABILITY, GOOD STRENGTH, BLEED RESISTANCE, MIGRATION RESISTANCE, AND LOW OR NO TOXICITY ENGELHARD CORPORATION 2004-06-29 US disclosed
EP-1104444-B1 STRONG GREEN-SHADE YELLOW DISAZO PIGMENT ENGELHARD CORP (US) 2002-12-18 EP disclosed
US-6254671-B1 Very green-shade yellow metallized disazo pigment ENGELHARD CORPORATION 2001-07-03 US disclosed
EP-1104444-A1 STRONG GREEN-SHADE YELLOW DISAZO PIGMENT Engelhard Corporation (US) 2001-06-06 EP disclosed
WO-2000009614-A1 STRONG GREEN-SHADE YELLOW DISAZO PIGMENT ENGELHARD CORPORATION (US) 2000-02-24 WO disclosed
US-5889162-A COUPLING A DIAZONIUM COMPONENT MADE FROM ONE OR MORE AROMATIC AMINES SUCH AS 2-ETHOXYANILINE WITH AT LEAST ONE COUPLING AGENT; SUITABLE FOR USE IN PLASTICS, PAINTS AND INKS ENGELHARD CORPORATION (US) 1999-03-30 US disclosed
EP-0025164-B1 DISAZO COMPOUNDS, PROCESS FOR THEIR PREPARATION AND USE HOECHST AKTIENGESELLSCHAFT (DE) 1983-04-13 EP disclosed
EP-0025164-A1 Disazo compounds, process for their preparation and use HOECHST AKTIENGESELLSCHAFT (DE) 1981-03-18 EP disclosed