SCHEMBL2909834

SCHEMBL2909834

CCc1ccc(-c2cn(CCCNc3ccc([N+](=O)[O-])c(N)n3)cc2NC(=O)CN2CC[C@H](N(C)C)C2)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
RECQL P46063 1/20 0.33
KDR P35968 1/20 0.33
GRM2 Q14416 1/20 0.33
MAPK1 P28482 1/20 0.33
GSK3B P49841 2/20 0.32
GSK3A P49840 1/20 0.32
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
KCNH2 Q12809 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
JAK2 O60674 1/20 0.31
AXL P30530 1/20 0.31
MERTK Q12866 1/20 0.31
HDAC1 Q13547 1/20 0.31
TLR7 Q9NYK1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910867 1.00 ALDH1A1 (0.33) ALDH1A1POLBLMNARECQLKDR
SCHEMBL2912942 0.89 ALDH1A1 (0.35) ALDH1A1POLBLMNARECQLGRM2
SCHEMBL2910392 0.89 ALDH1A1 (0.35) ALDH1A1POLBLMNARECQLGRM2
SCHEMBL2913211 0.89 POLB (0.46) ALDH1A1POLBRECQLMAPK1GSK3B
SCHEMBL2903975 0.89 POLB (0.39) ALDH1A1POLBRECQLMAPK1GSK3B
SCHEMBL2907498 0.88 RAB9A (0.38) ALDH1A1POLBLMNARECQLMAPK1
SCHEMBL2904881 0.88 RAB9A (0.39) ALDH1A1LMNAMAPK1GSK3BGSK3A
SCHEMBL2904441 0.87 ALDH1A1 (0.35) ALDH1A1POLBLMNARECQLMAPK1
SCHEMBL2910394 0.87 KDM4E (0.39) ALDH1A1POLBLMNAMAPK1GSK3B
SCHEMBL2911693 0.86 GSK3B (0.45) ALDH1A1POLBLMNARECQLKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed