SCHEMBL2912772

SCHEMBL2912772

CCOc1cc2nc(CC)c(C(=O)O)c(Nc3ccc(F)c(Cl)c3)c2cc1N1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
EGFR P00533 14/20 0.42
EPHA2 P29317 1/20 0.42
KDR P35968 1/20 0.42
EPHB4 P54760 1/20 0.42
ERBB2 P04626 4/20 0.41
FBP1 P09467 1/20 0.39
CSF1R P07333 2/20 0.39
KCNH2 Q12809 2/20 0.39
SCN5A Q14524 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913781 0.87 KCNH2 (0.47) EGFRCSF1RKCNH2SCN5A
SCHEMBL2907522 0.87 CSF1R (0.48) MAPTEGFRERBB2FBP1CSF1R
SCHEMBL2911203 0.83 CSF1R (0.56) MAPTEGFREPHA2KDREPHB4
SCHEMBL2912768 0.82 CA2 (0.51) MAPTEGFRERBB2CSF1RKCNH2
SCHEMBL27765555 0.80 EGFR (0.44) MAPTEGFRERBB2CSF1RKCNH2
SCHEMBL2911700 0.79 KCNH2 (0.51) MAPTEGFRKDRFBP1CSF1R
SCHEMBL2913426 0.79 CSF1R (0.51) CSF1RKCNH2SCN5A
SCHEMBL2908706 0.78 KCNH2 (0.46) MAPTEGFRKDRCSF1RKCNH2
SCHEMBL2910817 0.75 CSF1R (0.63) EGFRCSF1RKCNH2SCN5A
SCHEMBL2905929 0.74 CSF1R (0.53) EPHA2KDREPHB4ERBB2CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed