SCHEMBL2913405

SCHEMBL2913405

Cc1c(O[Si](C)(C)C(C)(C)C)cccc1B(O)O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.39
ORAI1 Q96D31 1/20 0.34
ORAI2 Q96SN7 1/20 0.34
ORAI3 Q9BRQ5 1/20 0.34
LIPE Q05469 1/20 0.33
DRD2 P14416 1/20 0.31
PREP P48147 1/20 0.31
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15269311 0.84 ENPP2 (0.52) ENPP2ORAI1ORAI2ORAI3LIPE
SCHEMBL21751366 0.82 ENPP2 (0.38) ENPP2ORAI1ORAI2ORAI3LIPE
SCHEMBL16501188 0.79 MAPT (0.42)
SCHEMBL2555302 0.79 DRD2 (0.33) DRD2PREP
SCHEMBL2905195 0.77 PREP (0.33) DRD2PREP
SCHEMBL17621111 0.76 CYP2D6 (0.33) PREP
SCHEMBL7247912 0.76 TSHR (0.45) PREP
SCHEMBL2367203 0.75 CA12 (0.34) DRD2PREP
SCHEMBL25400416 0.75 DRD2 (0.33) DRD2PREP
SCHEMBL16456193 0.75 PDCD1 (0.41) DRD2PREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100267775-A1 OXADIAZOLIDINEDIONE COMPOUND ASTELLAS PHARMA INC. (JP) 2010-10-21 US disclosed
EP-2216330-A1 OXADIAZOLIDINEDIONE COMPOUND Astellas Pharma Inc. (JP) 2010-08-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100267775-A1 OXADIAZOLIDINEDIONE COMPOUND GPR119, GLP1R, GPR4 ENPP2 1501/4885ORAI1 268/4885ORAI2 506/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.