SCHEMBL29136197

SCHEMBL29136197

COc1ccc2c(c[c]n2Cc2ccc(F)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
LMNA P02545 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
CYP2C19 P33261 1/20 0.44
BLM P54132 1/20 0.44
PMP22 Q01453 1/20 0.44
MAPT P10636 3/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR1A P08908 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
MAOB P27338 1/20 0.40
P2RX7 Q99572 2/20 0.40
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29136196 0.92 MAPT (0.43) KDM4ELMNACYP2C9TSHRMAPT
SCHEMBL29136185 0.82 CCR2 (0.52) KDM4EMAPTALDH1A1POLBKMT2A
SCHEMBL29136191 0.80 MAPT (0.40) MAPTHTR3EHTR3BHTR1AHTR3A
SCHEMBL28995440 0.79 CYP19A1 (0.40) KDM4ELMNANPSR1MAPTHTR1A
SCHEMBL3091129 0.77 P2RX4 (0.48) KDM4ELMNANPSR1MAPTHTR3A
SCHEMBL29136199 0.76 CCR2 (0.55) KDM4ELMNACYP1A2CYP3A4CYP2C9
SCHEMBL5894379 0.76 HDAC8 (0.56) KDM4ELMNANPSR1CYP1A2CYP3A4
SCHEMBL29136188 0.75 RAB9A (0.42) KDM4ELMNANPSR1TSHRMAPT
SCHEMBL28415278 0.74 DCTPP1 (0.41) KDM4ELMNAMAPTALDH1A1SMN1; SMN2
SCHEMBL29136202 0.71 KMT2A (0.55) KDM4ELMNATSHRMAPTHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117003739-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 安徽中医药大学 2023-11-07 CN disclosed