SCHEMBL29136750

SCHEMBL29136750

CNC(=O)Oc1ncccc1C(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
P2RY1 P47900 14/20 0.45
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
P2RY14 Q15391 2/20 0.43
PLCG1 P19174 1/20 0.40
ALOX5 P09917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29100772 0.81 P2RY1 (0.44) P2RY1P2RY14PLCG1
SCHEMBL21121867 0.75 KMT2A (0.50) ALDH1A1CHRM2CHRM4CHRM5CHRM1
SCHEMBL5566828 0.75 ALDH1A1 (0.45) ALDH1A1
SCHEMBL10550352 0.74 ALDH1A1 (0.50) ALDH1A1CHRM2CHRM4CHRM5CHRM1
SCHEMBL77829 0.73 ALDH1A1 (0.56) ALDH1A1CHRM2CHRM4CHRM5CHRM1
SCHEMBL21122068 0.73 BACE1 (0.42) ALDH1A1CHRM2CHRM4CHRM5CHRM1
Bromide SCHEMBL6851419 0.72 ALDH1A1 (0.54) ALDH1A1CHRM2CHRM4CHRM5CHRM1
SCHEMBL14803765 0.72 PLK1 (0.43) ALDH1A1P2RY1PLCG1
SCHEMBL77689 0.72 SLC22A12 (0.46) P2RY1P2RY14PLCG1
SCHEMBL6022886 0.71 NLRP3 (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed