SCHEMBL29136858

SCHEMBL29136858

C=CC(=O)Oc1c(Br)ccc(OC)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.40
ALDH1A1 P00352 2/20 0.38
THRB P10828 2/20 0.36
TSHR P16473 1/20 0.36
APOBEC3A P31941 1/20 0.36
HTT P42858 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
KDM4E B2RXH2 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TUBB1 Q9H4B7 2/20 0.35
PTGS1 P23219 1/20 0.35
ABL1 P00519 1/20 0.35
RIN1 Q13671 1/20 0.35
TNFRSF1A P19438 1/20 0.35
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28525364 0.85 ERN1 (0.50) ERN1ALDH1A1THRBTSHRAPOBEC3A
SCHEMBL15239366 0.80 MEN1 (0.43) THRBKDM4ETUBB1KMT2AHPGD
SCHEMBL3676845 0.78 THRB (0.39) ERN1ALDH1A1THRBKDM4ERXFP1
SCHEMBL28783574 0.77 TSHR (0.43) ERN1ALDH1A1TSHRAPOBEC3AHTT
SCHEMBL30406222 0.76 ALDH1A1 (0.53) ALDH1A1THRBKDM4ETUBB1PTGS1
SCHEMBL27368124 0.76 ACHE (0.50) ERN1ALDH1A1HTTKDM4ETUBB1
SCHEMBL29135178 0.75 PTPN1 (0.42) ERN1ALDH1A1THRBKDM4ERXFP1
SCHEMBL147312 0.74 TUBB1 (0.46) ERN1ALDH1A1TSHRAPOBEC3AHTT
SCHEMBL24810564 0.74 NFE2L2 (0.47) ERN1ALDH1A1THRBKDM4EKMT2A
SCHEMBL28295437 0.74 ABCG2 (0.45) ALDH1A1THRBKDM4ETUBB1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed