SCHEMBL29136924

SCHEMBL29136924

COc1ccnc(/C=C/C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.51
ATM Q13315 1/20 0.51
KDM4E B2RXH2 6/20 0.48
MAPK1 P28482 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
CCR1 P32246 1/20 0.46
CCR5 P51681 1/20 0.46
CCR8 P51685 1/20 0.46
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
ALOX15 P16050 1/20 0.44
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 2/20 0.42
SNCA P37840 2/20 0.42
PKM P14618 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2830915 0.86 CCR1 (0.44) KDM4EMAPK1NPSR1CCR1CCR5
SCHEMBL29879467 0.86 CCR1 (0.44) KDM4EMAPK1NPSR1CCR1CCR5
SCHEMBL2830917 0.86 CCR1 (0.44) KDM4EMAPK1NPSR1CCR1CCR5
SCHEMBL12501426 0.83 PTGS2 (0.44) KDM4EMAPK1NPSR1CCR1CCR5
SCHEMBL2956493 0.78 SMN1; SMN2 (0.42) THRBKDM4ENPSR1CCR1CCR5
SCHEMBL2956488 0.78 SMN1; SMN2 (0.42) THRBKDM4ENPSR1CCR1CCR5
SCHEMBL9756904 0.78 ALDH1A1 (0.63) THRBKDM4EALDH1A1SMN1; SMN2LMNA
SCHEMBL9756901 0.78 ALDH1A1 (0.63) THRBKDM4EALDH1A1SMN1; SMN2LMNA
SCHEMBL1124202 0.77 THRB (0.59) THRBATMKDM4EMAPK1ALDH1A1
SCHEMBL5664366 0.77 PLAU (0.50) KDM4EMAPK1NPSR1CCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed