SCHEMBL29137229

SCHEMBL29137229

Cc1ccccc1CN1CCN(c2cc(=O)n(C)c3ccc(Cl)nc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPC5 Q9UL62 4/20 0.48
KDM4E B2RXH2 2/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 3/20 0.45
MAPT P10636 2/20 0.45
TNKS O95271 1/20 0.43
PARP1 P09874 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
KMT2A Q03164 2/20 0.42
RAB9A P51151 2/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.40
PLA2G1B P04054 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
HTR7 P34969 1/20 0.40
HTR1A P08908 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
CNR1 P21554 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30616732 0.87 KDM4E (0.46) KDM4ELMNAMAPTTNKSPARP1
SCHEMBL30616746 0.85 GRM2 (0.41) KDM4ELMNAMAPTTNKSPARP1
SCHEMBL29137184 0.84 DRD2 (0.40) LMNATP53MAPTALDH1A1
SCHEMBL28549345 0.84 KDM4E (0.48) KDM4ELMNATP53MAPTALDH1A1
SCHEMBL29137205 0.83 ALDH1A1 (0.49) KDM4ELMNAMAPTKMT2AMEN1
SCHEMBL30616705 0.83 TRPC5 (0.39) TRPC5KDM4EALDH1A1HTR1AHTR1D
SCHEMBL30616722 0.82 GRM2 (0.44) TRPC5KDM4ELMNAMAPTPARP1
SCHEMBL30616712 0.82 GRM2 (0.44) TRPC5KDM4EPARP1ALDH1A1HTR1A
SCHEMBL30616730 0.82 ALDH1A1 (0.46) TRPC5KDM4EMAPTALDH1A1COMT
SCHEMBL29137283 0.81 DRD4 (0.38) MAPTKMT2AMEN1ALDH1A1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112585139-B Naphthyridinone compounds as T cell activators 百时美施贵宝公司 2023-12-01 CN disclosed