SCHEMBL2914288

SCHEMBL2914288

CC(C)(C)Nc1nc(N)c(F)cc1F

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 10/20 0.35
CCNE2 O96020 9/20 0.35
CCNE1 P24864 9/20 0.35
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
HTT P42858 1/20 0.34
CCNA2 P20248 1/20 0.33
CCNA1 P78396 1/20 0.33
KHK P50053 1/20 0.33
CDK4 P11802 4/20 0.33
CCND1 P24385 4/20 0.33
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GLP1R P43220 1/20 0.32
LATS1 O95835 3/20 0.31
LATS2 Q9NRM7 2/20 0.31
BCDIN3D Q7Z5W3 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alcohol SCHEMBL27466006 0.92 SLC29A1 (0.33) CDK2CCNE2CCNE1LMNAPOLB
SCHEMBL7170682 0.84 GLP1R (0.39) CDK2CCNE2CCNE1LMNAPOLB
SCHEMBL7172045 0.80 LMNA (0.36) CDK2CCNE2CCNE1LMNAPOLB
SCHEMBL7859690 0.80 KHK (0.45) CDK2CCNE2CCNE1LMNAHTT
SCHEMBL7168981 0.78 KHK (0.36) LMNAKHKMAPTSMN1; SMN2
SCHEMBL7169151 0.73 CDK2 (0.36) CDK2CCNE2CCNE1LMNAPOLB
SCHEMBL7171751 0.73 APP (0.38) KHKGLP1R
SCHEMBL7169449 0.72 BCL6 (0.56) CDK2LMNAPOLBHTTLATS1
SCHEMBL7859660 0.72 GLP1R (0.41) CDK2CCNE2CCNE1LMNAPOLB
SCHEMBL1565794 0.71 KHK (0.46) LMNAKHKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1813610-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF WAKUNAGA PHARMA CO LTD (JP) 2010-09-08 EP disclosed
US-7713997-B2 Pyridonecarboxylic acid derivatives or salts thereof WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2010-05-11 US disclosed
US-20090149440-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF WAKUNAGA PHARMACEUTICAL CO., LTD (JP) 2009-06-11 US disclosed
EP-1813610-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2007-08-01 EP disclosed
CN-1196683-C Amino-compound YUNAGA PHARMACEUTICAL CO LTD (JP) 2005-04-13 CN disclosed
US-6858625-B1 Quinolinecarboxylic acid derivative or salts thereof WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2005-02-22 US disclosed
CN-1136216-C Pyrone carboxylic acid derivate or its salt and antibiotic with the same as effective component ������ҩ��ʽ���� 2004-01-28 CN disclosed
EP-1193266-B1 QUINOLINECARBOXYLIC ACID DERIVATIVE OR SALTS THEREOF WAKUNAGA PHARMA CO LTD (JP) 2003-08-27 EP disclosed
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6586420-B1 Photostable bactericides WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2003-07-01 US disclosed
US-6156903-A Pyridonecarboxylic acid derivatives or their salts, and antibacterial agents containing the same as their effective components WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-12-05 US disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
US-6133284-A EXCELLENT BACTERICIDAL PROPERTIES AND ORAL ABSORPTION; INFECTIONS FROM GRAMNEGATIVE AND -POSITIVE BACTERIA; INTESTINAL ABSORPTION, METABOLIC STABILITY; SIDE EFFECT REDUCTION; NONPHOTOTOXICITY AND NONCYTOTOXICITY WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-17 US disclosed
CN-1258674-A Pyrone carboxylic acid derivate or its salt and antibiotic with the same as effective component YUNAGA PHARMACEUTICAL CO LTD (JP) 2000-07-05 CN disclosed
CN-1258672-A Amino-compound YUNAGA PHARMACEUTICAL CO LTD (JP) 2000-07-05 CN disclosed
EP-0992501-A2 Pyridonecarboxylic acid derivatives as antibacterial agents WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-04-12 EP disclosed
US-5998436-A Pyridonecarboxylic acid derivatives or their salts and antibacterial agent comprising the same as the active ingredient WAKUNAGA PHARMACEUTICALS CO., LTD. (JP) 1999-12-07 US disclosed
EP-0952151-A2 Intermediates for use in preparing novel pyridonecarboxylic acid derivatives or their salts WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-10-27 EP disclosed
EP-0911327-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR THEIR SALTS AND ANTIBACTERIAL AGENT COMPRISING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-04-28 EP disclosed
CN-1201459-A Novel pyridonecarboxylic acid derivative or salt thereof, and antibacterial agent containing same as active ingredient WAKUNAGA PHARMA CO LTD (JP) 1998-12-09 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090149440-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF SLC7A1, PLPBP, PYCR1 CDK2 1437/4885CCNE2 3675/4885CCNE1 2305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.