SCHEMBL2915261

SCHEMBL2915261

COc1cc(N)ccc1C(=O)NO.COc1ccc(N)cc1C(=O)NO

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
CRBN Q96SW2 1/20 0.48
HDAC8 Q9BY41 3/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
GAA P10253 3/20 0.44
CTSD P07339 1/20 0.44
PYGL P06737 1/20 0.43
HDAC11 Q96DB2 2/20 0.43
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GFER P55789 1/20 0.42
HSD17B10 Q99714 1/20 0.42
LMNA P02545 1/20 0.41
ALOX5 P09917 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL728419 0.94 ALDH1A1 (0.53) ALDH1A1HDAC8HDAC1HDAC6CYP1A2
SCHEMBL728203 0.94 ALDH1A1 (0.67) ALDH1A1CRBNGAACTSDPYGL
SCHEMBL5679153 0.81 ALDH1A1 (0.67) ALDH1A1CRBNHDAC1GAACTSD
SCHEMBL655826 0.81 ALDH1A1 (0.53) ALDH1A1CYP1A2CYP2C9CYP2C19GAA
SCHEMBL328279 0.81 ALDH1A1 (0.67) ALDH1A1CRBNGAACTSDPYGL
Hydrochloric Acid SCHEMBL2553196 0.80 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP2C9CYP2C19GAA
SCHEMBL13294935 0.79 HDAC7 (0.53) ALDH1A1CYP1A2CYP2C9CYP2C19GAA
SCHEMBL5925494 0.78 GAA (0.64) ALDH1A1CRBNGAACTSDPYGL
SCHEMBL570110 0.77 GAA (0.61) ALDH1A1GAAMAPTHSD17B10LMNA
SCHEMBL224165 0.77 ALDH1A1 (0.71) ALDH1A1CRBNGAAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222291-A2 COMPOUNDS FOR THE SELECTIVE TREATMENT OF THE INTESTINAL IMMUNO-INFLAMMATORY COMPONENT OF THE CELIAC DISEASE Giuliani International Limited (IE) 2010-09-01 EP claimed
WO-2009080828-A2 COMPOUNDS FOR THE SELECTIVE TREATMENT OF THE INTESTINAL IMMUNO-INFLAMMATORY COMPONENT OF THE CELIAC DISEASE GIULIANI INTERNATIONAL LIMITED (IE) 2009-07-02 WO claimed