SCHEMBL328279

SCHEMBL328279

CNC(=O)c1ccc(N)cc1OC

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.67
PLK1 P53350 1/20 0.53
CRBN Q96SW2 1/20 0.52
GAA P10253 5/20 0.49
MAPT P10636 2/20 0.49
HTT P42858 2/20 0.49
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.46
CTSD P07339 1/20 0.45
HSD17B1 P14061 1/20 0.45
PYGL P06737 1/20 0.44
PKM P14618 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TP53 P04637 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655826 0.86 ALDH1A1 (0.53) ALDH1A1PLK1GAAMAPTHTT
SCHEMBL5679153 0.86 ALDH1A1 (0.67) ALDH1A1CRBNGAAMAPTHTT
SCHEMBL728203 0.86 ALDH1A1 (0.67) ALDH1A1CRBNGAAMAPTHTT
Hydrochloric Acid SCHEMBL2553196 0.85 ALDH1A1 (0.51) ALDH1A1PLK1GAAMAPTHTT
SCHEMBL5925494 0.83 GAA (0.64) ALDH1A1CRBNGAAMAPTSMN1; SMN2
SCHEMBL224165 0.82 ALDH1A1 (0.71) ALDH1A1CRBNGAAMAPTHTT
SCHEMBL3850604 0.82 ALDH1A1 (0.61) ALDH1A1CRBNMAPTMAPK1SMN1; SMN2
SCHEMBL29530877 0.82 ALDH1A1 (0.61) ALDH1A1CRBNMAPTMAPK1SMN1; SMN2
SCHEMBL3110944 0.82 ALDH1A1 (0.61) ALDH1A1CRBNGAAMAPTHTT
SCHEMBL3850748 0.82 MAPT (0.63) ALDH1A1CRBNGAAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4640678-A1 NOVEL OXO-PYRIDINE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF Chengdu Shibeikang Biomedical Technology Co., Ltd. (CN) 2025-10-29 EP disclosed
CN-116082303-B Novel oxopyridines, intermediates and uses thereof 成都施贝康生物医药科技有限公司 2025-02-25 CN disclosed
WO-2024131841-A1 NOVEL OXO-PYRIDINE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF 成都施贝康生物医药科技有限公司 2024-06-27 WO disclosed
CN-116082303-A Novel oxopyridines, intermediates and uses thereof 成都施贝康生物医药科技有限公司 2023-05-09 CN disclosed
US-20230091047-A1 FUSED RING PYRIMIDONE DERIVATIVES FOR USE IN THE TREATMENT OF HBV INFECTION OR OF HBV-INDUCED DISEASES JANSSEN PHARMACEUTICA NV (BE) 2023-03-23 US disclosed
US-9913817-B2 Methods for preventing or reducing colon carcinogenesis NOGRA PHARMA LIMITED (IE) 2018-03-13 US disclosed
US-20180064667-A1 METHODS OF TREATING LACTOSE INTOLERANCE NOGRA PHARMA LTD (IE) 2018-03-08 US disclosed
US-20170056349-A1 Methods for Preventing or Reducing Colon Carcinogenesis NOGRA PHARMA LIMITED (IE) 2017-03-02 US disclosed
US-9487491-B2 Diamino heterocyclic carboxamide compound ASTELLAS PHARMA INC. (JP) 2016-11-08 US disclosed
EP-3009428-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND Astellas Pharma Inc. (JP) 2016-04-20 EP disclosed
US-20140371196-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND ASTELLAS PHARMA INC. (JP) 2014-12-18 US disclosed
US-8501806-B2 Methods for preventing or reducing colon carcinogenesis NOGRA PHARMA LIMITED (IE) 2013-08-06 US disclosed
US-8138357-B2 Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field GIULIANI INTERNATIONAL LIMITED (IE) 2012-03-20 US disclosed
EP-2428508-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND Astellas Pharma Inc. (JP) 2012-03-14 EP disclosed
US-20120040968-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND WATERS TECHNOLOGIES CORPORATION (US) 2012-02-16 US disclosed
US-20110288058-A1 Methods for Preventing or Reducing Colon Carcinogenesis NOGRA PHARMA LIMITED (IE) 2011-11-24 US disclosed
US-20110288177-A1 Methods for Preventing or Reducing Colon Carcinogenesis NOGRA PHARMA LIMITED (IE) 2011-11-24 US disclosed
US-20110152225-A1 PPAR-Gamma Agonists for the Induction of Cationic Antimicrobial Peptide Expression as Immunoprotective Stimulants NOGRA PHARMA LIMITED (IE) 2011-06-23 US disclosed
WO-2010128659-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND アステラス製薬株式会社 (JP) 2010-11-11 WO disclosed
US-20090118357-A1 Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field GIULIANI INTERNATIONAL LIMITED (IE) 2009-05-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170056349-A1 Methods for Preventing or Reducing Colon Carcinogenesis NQO1, NFE2L2, CYBB ALDH1A1 103/4885PLK1 4308/4885CRBN 1306/4885
US-20230091047-A1 FUSED RING PYRIMIDONE DERIVATIVES FOR USE IN THE TREATMENT OF HBV INFECTION OR OF HBV-INDUCED DISEASES HAVCR2, HCCS, TYMP ALDH1A1 1508/4885PLK1 430/4885CRBN 4193/4885
US-20090118357-A1 Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field EGFR, ERBB3, FGFR3 ALDH1A1 2287/4885PLK1 3830/4885CRBN 704/4885
US-20140371196-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND EML4, ALK, ERBB4 ALDH1A1 1554/4885PLK1 1966/4885CRBN 1454/4885
US-20110288058-A1 Methods for Preventing or Reducing Colon Carcinogenesis NQO1, NFE2L2, CYBB ALDH1A1 103/4885PLK1 4308/4885CRBN 1306/4885
US-20110288177-A1 Methods for Preventing or Reducing Colon Carcinogenesis APC, GSTK1, GSTA1 ALDH1A1 126/4885PLK1 3854/4885CRBN 688/4885
US-20120040968-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND EML4, ALK, ERBB4 ALDH1A1 1554/4885PLK1 1966/4885CRBN 1454/4885
US-20180064667-A1 METHODS OF TREATING LACTOSE INTOLERANCE LCT, LPL, PPARG ALDH1A1 530/4885PLK1 3550/4885CRBN 4274/4885
US-20110152225-A1 PPAR-Gamma Agonists for the Induction of Cationic Antimicrobial Peptide Expression as Immunoprotective Stimulants PPARG, FABP2, PPARD ALDH1A1 983/4885PLK1 4399/4885CRBN 4784/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.