SCHEMBL29200055

SCHEMBL29200055

O=COCC(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.56
GSK3B P49841 2/20 0.56
ALDH1A1 P00352 1/20 0.54
MAPT P10636 1/20 0.54
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
MMP1 P03956 1/20 0.49
GRM4 Q14833 1/20 0.47
HSD11B1 P28845 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
SRD5A2 P31213 2/20 0.44
MMP2 P08253 1/20 0.44
MMP8 P22894 1/20 0.44
NR4A1 P22736 1/20 0.44
NR4A2 P43354 1/20 0.44
NR4A3 Q92570 1/20 0.44
PDPK1 O15530 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24239347 0.81 CES2 (0.56) ALDH1A1MAPTCES2SRD5A2
SCHEMBL20221553 0.80 MAPT (0.44) PTPN1GSK3BALDH1A1MAPTSRD5A2
SCHEMBL3391803 0.79 ALDH1A1 (0.60) PTPN1GSK3BALDH1A1MAPTCES2
SCHEMBL31423428 0.79 PTPN1 (0.59) PTPN1GSK3BALDH1A1MAPTCES2
SCHEMBL10465723 0.77 GSK3B (0.53) GSK3BALDH1A1MAPTCES2CES1
SCHEMBL17702639 0.77 NPC1 (0.53) GSK3BALDH1A1MAPTCES2CES1
SCHEMBL11074838 0.77 GSK3B (0.53) GSK3BALDH1A1MAPTCES2CES1
SCHEMBL28873117 0.77 PTPN1 (0.61) PTPN1GSK3BALDH1A1MAPTCES2
SCHEMBL20716307 0.76 VNN1 (0.43) HDAC8
SCHEMBL2865542 0.76 ALDH1A1 (0.70) PTPN1GSK3BALDH1A1MAPTCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed