SCHEMBL2925490

SCHEMBL2925490

Cc1cccc(C(=O)N2C[C@H]3C[C@H]3[C@H]2C(N)=O)c1-c1ccccc1F

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.37
MYC P01106 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HCRTR2 O43614 15/20 0.36
HCRTR1 O43613 14/20 0.36
PDE4B Q07343 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3415876 0.88 CDK4 (0.36) ALDH1A1HCRTR2HCRTR1PDE4B
SCHEMBL2925297 0.88 CDK4 (0.36) ALDH1A1HCRTR2HCRTR1PDE4B
SCHEMBL2924242 0.86 FABP4 (0.42) PIK3CDMYCALDH1A1HCRTR2HCRTR1
SCHEMBL2931912 0.86 APOB (0.38) PIK3CDALDH1A1HCRTR2HCRTR1
SCHEMBL2925493 0.85 HCRTR2 (0.37) PIK3CDMYCHCRTR2HCRTR1
SCHEMBL2928147 0.85 HCRTR1 (0.36) PIK3CDALDH1A1HCRTR2HCRTR1
SCHEMBL2931039 0.84 HCRTR2 (0.39) PIK3CDHCRTR2HCRTR1PDE4B
SCHEMBL2928983 0.83 GRM2 (0.40) HCRTR2HCRTR1PDE4B
SCHEMBL2932481 0.83 GRM2 (0.40) HCRTR2HCRTR1PDE4B
SCHEMBL2926433 0.81 MGLL (0.38) PIK3CDALDH1A1HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed