SCHEMBL2928147

SCHEMBL2928147

Cc1cc(-c2c(C)cccc2C(=O)N2C[C@H]3C[C@H]3[C@H]2C(N)=O)ccc1F

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.36
HCRTR2 O43614 11/20 0.36
CYP3A4 P08684 2/20 0.34
PIK3CD O00329 1/20 0.33
GRIN2B Q13224 1/20 0.33
PIK3CA P42336 1/20 0.33
CHRNA7 P36544 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ABL1 P00519 1/20 0.32
KIT P10721 1/20 0.32
FFAR1 O14842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2931039 0.88 HCRTR2 (0.39) HCRTR1HCRTR2PIK3CD
SCHEMBL2931912 0.88 APOB (0.38) HCRTR1HCRTR2PIK3CDALDH1A1
SCHEMBL2930073 0.86 PDE4B (0.37) HCRTR1HCRTR2
SCHEMBL2930954 0.86 POLB (0.39) HCRTR1HCRTR2PIK3CDPIK3CAALDH1A1
SCHEMBL2928151 0.86 HCRTR2 (0.35) HCRTR1HCRTR2CYP3A4GRIN2BFFAR1
SCHEMBL2925490 0.85 PIK3CD (0.37) HCRTR1HCRTR2PIK3CDALDH1A1
SCHEMBL2924242 0.85 FABP4 (0.42) HCRTR1HCRTR2PIK3CDPIK3CAALDH1A1
SCHEMBL2929656 0.84 HCRTR2 (0.37) HCRTR1HCRTR2CYP3A4GRIN2BPIK3CA
SCHEMBL2925366 0.84 HCRTR1 (0.39) HCRTR1HCRTR2CHRNA7
SCHEMBL2926251 0.84 HCRTR2 (0.39) HCRTR1HCRTR2PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed