SCHEMBL2925883

SCHEMBL2925883

Cc1ccc(C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)c(-c2cccc(C(C)C)c2)c1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.33
PDE10A Q9Y233 1/20 0.33
RXRA P19793 2/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
HCRTR2 O43614 6/20 0.32
HCRTR1 O43613 5/20 0.32
HDAC7 Q8WUI4 1/20 0.32
KRAS P01116 1/20 0.32
NR4A2 P43354 1/20 0.31
NOTUM Q6P988 2/20 0.31
CYP46A1 Q9Y6A2 1/20 0.31
ATM Q13315 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CTSA P10619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2924875 0.90 HCRTR2 (0.37) CHRM1HCRTR2HCRTR1HDAC7CYP46A1
SCHEMBL2926155 0.87 HDAC7 (0.43) HCRTR2HCRTR1HDAC7CYP46A1
SCHEMBL2929505 0.87 HCRTR2 (0.43) HCRTR2HCRTR1
SCHEMBL2925064 0.87 HCRTR2 (0.43) HCRTR2HCRTR1
SCHEMBL2930272 0.87 CHRM1 (0.46) CHRM1HCRTR2HCRTR1
SCHEMBL2925882 0.86 RXRA (0.33) CHRM1PDE10ARXRARXRBRXRG
SCHEMBL2931139 0.85 HCRTR1 (0.39) HCRTR2HCRTR1
SCHEMBL2924236 0.85 KDM1A (0.35) HCRTR2HCRTR1HDAC7CYP46A1
SCHEMBL2933414 0.84 HCRTR1 (0.38) HCRTR2HCRTR1
SCHEMBL2926961 0.82 MEN1 (0.43) HCRTR2HCRTR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed