SCHEMBL29266142

SCHEMBL29266142

CN(CCCO)C(=O)c1ccc(N2CCCN(C(=O)O)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
HRH3 Q9Y5N1 2/20 0.41
AKR1C3 P42330 1/20 0.39
PDK2 Q15119 1/20 0.38
MAPT P10636 3/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
STAT1 P42224 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
DRD4 P21917 1/20 0.37
ESRRB O95718 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22291069 0.84 TMEM97 (0.46) HRH3MAPTLMNAKMT2AMEN1
SCHEMBL22291101 0.80 ALDH1A1 (0.45) ALDH1A1PDK2TSHRHSD17B10ESRRB
SCHEMBL22291198 0.78 CDK8 (0.42) ALDH1A1PDK2NPC1DRD4
SCHEMBL24399377 0.76 ALDH1A1 (0.35) ALDH1A1HRH3MAPTTSHRKMT2A
SCHEMBL22291202 0.73 CDK8 (0.50) ALDH1A1HRH3MAPTHPGDRAB9A
SCHEMBL30988055 0.73 CDK8 (0.50) ALDH1A1HRH3MAPTHPGDRAB9A
SCHEMBL64400 0.72 ALDH1A1 (0.57) ALDH1A1AKR1C3MAPTNPC1LMNA
SCHEMBL25417126 0.71 ALDH1A1 (0.43) ALDH1A1MAPTTSHRHSD17B10ESRRB
SCHEMBL25415646 0.71 SIGMAR1 (0.42) ALDH1A1HRH3PDK2MAPTLMNA
SCHEMBL18641154 0.70 DRD2 (0.52) ALDH1A1MAPTDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677341-B Bicyclic pyridine compositions and methods for their use in cancer treatment 南卡罗莱纳大学 2024-07-05 CN disclosed
CN-113677341-A Bicyclic pyridine compositions and methods of use for cancer treatment 南卡罗莱纳大学 2021-11-19 CN disclosed