SCHEMBL29280467

SCHEMBL29280467

C[Si](C)(C)CCOCn1cc(-c2ccncc2)c(-c2ccc(O)cc2)n1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.44
SLC6A3 Q01959 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PDE10A Q9Y233 3/20 0.41
MAPK3 P27361 1/20 0.41
MAPK1 P28482 1/20 0.41
MAPK13 O15264 1/20 0.40
CSNK1D P48730 1/20 0.40
CSNK1E P49674 1/20 0.40
MAPK12 P53778 1/20 0.40
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24951243 0.85 BRAF (0.43) BRAFSLC6A3MEN1KMT2APDE10A
SCHEMBL24950801 0.83 PDE10A (0.51) SLC6A3PDE10A
SCHEMBL31074565 0.80 MAPK14 (0.34) BRAFSLC6A3MEN1KMT2APDE10A
SCHEMBL31111573 0.80 DGAT1 (0.37) BRAFSLC6A3PDE10AMAPK3MAPK1
SCHEMBL24950777 0.79 BRAF (0.57) BRAFSLC6A3MEN1KMT2AMAPK3
SCHEMBL1847543 0.79 BRAF (0.39) BRAFSLC6A3PDE10AMAPK3MAPK1
SCHEMBL1847873 0.79 TGFBR1 (0.39) BRAFSLC6A3PDE10AMAPK14
SCHEMBL1846834 0.78 BRAF (0.37) BRAFSLC6A3PDE10AMAPK3MAPK1
SCHEMBL31111773 0.77 PDE10A (0.37) PDE10AMAPK13CSNK1DCSNK1EMAPK12
SCHEMBL1758620 0.77 BRAF (0.46) BRAFSLC6A3MEN1KMT2APDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117751107-A Organic pyridine-pyrazole compounds and uses thereof 博善人工智能剑桥有限公司 2024-03-22 CN disclosed