SCHEMBL2928151

SCHEMBL2928151

Cc1cc(-c2c(C)cccc2C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)ccc1F

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 17/20 0.35
HCRTR1 O43613 16/20 0.35
CYP3A4 P08684 2/20 0.35
FFAR1 O14842 1/20 0.35
GRIN2B Q13224 1/20 0.34
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2931914 0.90 HCRTR2 (0.39) HCRTR2HCRTR1
SCHEMBL2931040 0.89 HCRTR2 (0.40) HCRTR2HCRTR1
SCHEMBL2930074 0.87 SLC6A7 (0.35) HCRTR2HCRTR1
SCHEMBL2930955 0.86 HCRTR2 (0.38) HCRTR2HCRTR1
SCHEMBL2928147 0.86 HCRTR1 (0.36) HCRTR2HCRTR1CYP3A4FFAR1GRIN2B
SCHEMBL2924244 0.85 CYP46A1 (0.39) HCRTR2HCRTR1
SCHEMBL2925368 0.84 HCRTR1 (0.41) HCRTR2HCRTR1GRIN2B
SCHEMBL2925493 0.84 HCRTR2 (0.37) HCRTR2HCRTR1
SCHEMBL2930216 0.83 TP53 (0.39)
SCHEMBL2929658 0.83 HCRTR2 (0.36) HCRTR2HCRTR1CYP3A4GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed