SCHEMBL2928252

SCHEMBL2928252

NC(=O)Nc1sc(-c2ccc(CN3CCOCC3)c(F)c2)cc1OC(N)=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.42
JAK2 O60674 3/20 0.40
KCNH2 Q12809 2/20 0.40
SCN9A Q15858 3/20 0.40
JAK3 P52333 1/20 0.39
MOK Q9UQ07 4/20 0.39
IKBKE Q14164 1/20 0.38
BDKRB1 P46663 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
MEN1 O00255 1/20 0.38
IKBKB O14920 1/20 0.38
EIF2AK2 P19525 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CYP2A13 Q16696 1/20 0.37
KCNJ1 P48048 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2933735 0.89 CHEK1 (0.44) CHEK1JAK2KCNH2SCN9AJAK3
SCHEMBL1928063 0.86 CHEK1 (0.58) CHEK1JAK2KCNH2JAK3MEN1
SCHEMBL2934362 0.85 CHEK1 (0.58) CHEK1JAK2KCNH2JAK3MEN1
SCHEMBL2932975 0.83 PTGER1 (0.43) CHEK1JAK2KCNH2SCN9AJAK3
SCHEMBL2932197 0.83 CHEK1 (0.48) CHEK1JAK2KCNH2JAK3IKBKB
SCHEMBL5243288 0.83 CHEK1 (0.41) CHEK1JAK2KCNH2JAK3IKBKE
SCHEMBL2931062 0.82 CHEK1 (0.59) CHEK1JAK2KCNH2JAK3IKBKB
SCHEMBL2925535 0.82 JAK2 (0.43) CHEK1JAK2KCNH2JAK3IKBKE
SCHEMBL2930060 0.76 CHEK1 (0.70) CHEK1JAK2MEN1IKBKBEIF2AK2
SCHEMBL2927139 0.76 CHEK1 (0.41) CHEK1JAK2KCNH2JAK3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421074-B1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2010-09-29 EP claimed