SCHEMBL5243288

SCHEMBL5243288

NC(=O)Nc1sc(-c2ccc3sc(CN4CCOCC4)cc3c2)cc1OC(N)=O

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.41
MCHR1 Q99705 1/20 0.41
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40
KCNH2 Q12809 1/20 0.40
S1PR5 Q9H228 1/20 0.38
CD274 Q9NZQ7 1/20 0.37
CA2 P00918 4/20 0.37
TBK1 Q9UHD2 2/20 0.37
FAAH O00519 1/20 0.37
WNT1 P04628 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
IKBKE Q14164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5210487 0.86 CHEK1 (0.57) CHEK1MCHR1JAK2JAK3KCNH2
SCHEMBL2934362 0.85 CHEK1 (0.58) CHEK1JAK2JAK3KCNH2TBK1
SCHEMBL2933735 0.83 CHEK1 (0.44) CHEK1JAK2JAK3KCNH2
SCHEMBL2928252 0.83 CHEK1 (0.42) CHEK1JAK2JAK3KCNH2IKBKE
SCHEMBL2932197 0.82 CHEK1 (0.48) CHEK1JAK2JAK3KCNH2FAAH
SCHEMBL2925535 0.81 JAK2 (0.43) CHEK1JAK2JAK3KCNH2TBK1
SCHEMBL2931062 0.81 CHEK1 (0.59) CHEK1JAK2JAK3KCNH2TBK1
SCHEMBL2932975 0.79 PTGER1 (0.43) CHEK1JAK2JAK3KCNH2
SCHEMBL2930060 0.76 CHEK1 (0.70) CHEK1JAK2TBK1
SCHEMBL2927139 0.76 CHEK1 (0.41) CHEK1JAK2JAK3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421079-B1 THIOPHENYL COMPOUNDS AS MEDICAMENTS ASTRAZENECA AB (SE) 2007-02-07 EP claimed