SCHEMBL29285186

SCHEMBL29285186

Cc1ccc(S(=O)(=O)n2c(-c3cnn(CC4CCOCC4)c3)cc3c(Cl)c(C#N)cnc32)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
IKBKE Q14164 2/20 0.34
TBK1 Q9UHD2 2/20 0.34
AXL P30530 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
TTK P33981 1/20 0.33
RET P07949 3/20 0.33
LRRK2 Q5S007 2/20 0.33
FGFR1 P11362 3/20 0.33
FGFR3 P22607 3/20 0.33
KDR P35968 3/20 0.33
FGFR4 P22455 2/20 0.33
TYRO3 Q06418 1/20 0.33
FGFR2 P21802 1/20 0.33
FLT3 P36888 1/20 0.33
EED O75530 1/20 0.32
RBBP4 Q09028 1/20 0.32
SUZ12 Q15022 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29285182 0.83 CCNA2 (0.37) PIK3CDPTGDR2LRRK2CDK2
SCHEMBL15586787 0.75 MAOA (0.39) PTGDR2LRRK2
SCHEMBL30877298 0.72 RAPGEF4 (0.40) PIK3CDPIK3CAAXLTTKLRRK2
SCHEMBL1354815 0.71 CDK2 (0.39) LRRK2FLT3CCNT1CDK1CCNB1
SCHEMBL1356338 0.71 CDK2 (0.39) PTGDR2KDRCCNT1CDK1CCNB1
SCHEMBL30877369 0.70 ALDH1A1 (0.37) PTGDR2LRRK2
SCHEMBL29285155 0.70 ALDH1A1 (0.37) PTGDR2LRRK2
SCHEMBL29285170 0.70 PTGDR2 (0.41) PTGDR2RET
SCHEMBL30877398 0.67 TTK (0.35) TTK
SCHEMBL28569194 0.67 BTK (0.42) PTGDR2LRRK2FLT3CCNT1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964643-B Pyrrole [2,3-b ] pyridine derivative and preparation method and application thereof 苏州朗睿生物医药有限公司 2024-07-02 CN disclosed
CN-117964643-A Pyrrole [2,3-b ] pyridine derivative and preparation method and application thereof 苏州朗睿生物医药有限公司 2024-05-03 CN disclosed