SCHEMBL2929133

SCHEMBL2929133

Cc1ccc(C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)c(-c2cccc(OC(F)(F)F)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 9/20 0.40
HCRTR2 O43614 9/20 0.40
PIM1 P11309 5/20 0.40
PIM2 Q9P1W9 5/20 0.40
MMP2 P08253 1/20 0.38
MMP3 P08254 1/20 0.38
CFD P00746 2/20 0.38
DGAT2 Q96PD7 1/20 0.37
PDE10A Q9Y233 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2931139 0.89 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL2924875 0.87 HCRTR2 (0.37) HCRTR1HCRTR2
SCHEMBL2929132 0.87 HCRTR1 (0.42) HCRTR1HCRTR2PIM1PIM2MMP2
SCHEMBL2933414 0.86 HCRTR1 (0.38) HCRTR1HCRTR2
SCHEMBL2925423 0.86 CFD (0.40) HCRTR1HCRTR2PIM1PIM2MMP2
SCHEMBL2925064 0.85 HCRTR2 (0.43) HCRTR1HCRTR2
SCHEMBL2929505 0.85 HCRTR2 (0.43) HCRTR1HCRTR2
SCHEMBL2926155 0.84 HDAC7 (0.43) HCRTR1HCRTR2
SCHEMBL2930272 0.83 CHRM1 (0.46) HCRTR1HCRTR2
SCHEMBL2925883 0.82 CHRM1 (0.33) HCRTR1HCRTR2PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed