SCHEMBL2929672

SCHEMBL2929672

COc1ncnc2sc(NC(=O)ON3CCN(C(=O)c4ccc(C(F)(F)F)nc4)CC3)nc12

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.36
PIK3CD O00329 4/20 0.35
PIK3R1 P27986 3/20 0.35
SFRP1 Q8N474 1/20 0.35
MAPK7 Q13164 2/20 0.34
TRPV1 Q8NER1 1/20 0.34
LRRK2 Q5S007 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
ADORA2A P29274 2/20 0.34
ADORA2B P29275 2/20 0.34
ADORA1 P30542 2/20 0.34
EPHX2 P34913 1/20 0.34
STAT3 P40763 3/20 0.33
PIK3CG P48736 1/20 0.33
ITK Q08881 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1761050 0.90 HPGDS (0.40) KCNH2SFRP1MAPK7TRPV1LRRK2
SCHEMBL2931313 0.86 LRRK2 (0.38) KCNH2PIK3CDMAPK7LRRK2ADORA2A
SCHEMBL2932134 0.85 PPARD (0.42) KCNH2PIK3CDPIK3R1PIK3CG
SCHEMBL2927299 0.81 PIK3CG (0.36) PIK3CDPIK3R1ADORA2AADORA2BADORA1
SCHEMBL2931856 0.80 ALDH1A1 (0.44) ADORA2AADORA1
SCHEMBL2929996 0.77 PKLR (0.38) KCNH2TRPV1ADORA2AADORA2BADORA1
SCHEMBL1761042 0.76 PPARD (0.43)
SCHEMBL3041508 0.76 PHGDH (0.47) ADORA2A
SCHEMBL2932276 0.76 CYP2D6 (0.41) TRPV1ADORA2AADORA2BADORA1
SCHEMBL1761048 0.75 HPGDS (0.44) KCNH2PIK3CDMAPK7LRRK2PIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed