SCHEMBL29315909

SCHEMBL29315909

COC(=O)Cc1c(-c2cn[nH]c2)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 0.46
ROCK1 Q13464 19/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29315913 0.87 ROCK1 (0.39) ROCK2ROCK1
SCHEMBL29314121 0.77 POLQ (0.44) ROCK2ROCK1
SCHEMBL31009206 0.75 ROCK2 (0.36) ROCK2
SCHEMBL29316278 0.74 NPBWR1 (0.39) ROCK2ROCK1
SCHEMBL29315906 0.73 NOTUM (0.47)
SCHEMBL31648382 0.68 POLQ (0.56)
SCHEMBL29316276 0.65 ROCK2 (0.39) ROCK2ROCK1
SCHEMBL1296063 0.65 HSP90AB1 (0.56)
SCHEMBL31009157 0.64 POLQ (0.46) ROCK2ROCK1
SCHEMBL14661309 0.64 P2RX7 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed