SCHEMBL29316655

SCHEMBL29316655

NNC(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.42
P2RX1 P51575 8/20 0.41
P2RX7 Q99572 4/20 0.41
P2RX4 Q99571 3/20 0.40
NR5A2 O00482 1/20 0.40
NR5A1 Q13285 1/20 0.40
TMPRSS4 Q9NRS4 1/20 0.40
P2RX3 P56373 1/20 0.39
ALDH1A1 P00352 3/20 0.39
ATM Q13315 1/20 0.39
GFER P55789 1/20 0.39
GAA P10253 3/20 0.38
MAPT P10636 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
KDM4E B2RXH2 1/20 0.38
NSD2 O96028 1/20 0.38
LMNA P02545 1/20 0.38
ALPL P05186 1/20 0.38
POLB P06746 1/20 0.38
ALPI P09923 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14880120 0.81 CES2 (0.50) CES2P2RX1P2RX7P2RX4ALDH1A1
SCHEMBL25574138 0.79 CES2 (0.47) CES2ALDH1A1KDM4E
SCHEMBL5220850 0.78 CES2 (0.66) CES2TMPRSS4ALDH1A1ATMGAA
SCHEMBL10577013 0.77 NR5A2 (0.65) NR5A2NR5A1ALDH1A1GFERGAA
SCHEMBL29316641 0.77 NOTUM (0.51) CES2P2RX1TMPRSS4GFERGAA
SCHEMBL29316976 0.74 ALDH1A1 (0.48) CES2TMPRSS4ALDH1A1MAPTMEN1
SCHEMBL391593 0.73 CES2 (0.45) CES2ALDH1A1POLB
SCHEMBL10524850 0.71 ALDH1A1 (0.61) CES2P2RX1P2RX7P2RX4TMPRSS4
SCHEMBL24209801 0.71 ALDH1A1 (0.53) CES2P2RX1ALDH1A1ATMKDM4E
SCHEMBL3277286 0.71 GAA (0.61) CES2P2RX1ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed