SCHEMBL29316976

SCHEMBL29316976

NNC(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1O

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
GPR35 Q9HC97 4/20 0.40
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA9 Q16790 3/20 0.39
TMPRSS4 Q9NRS4 1/20 0.39
MAPT P10636 1/20 0.38
CHRNA7 P36544 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
CES2 O00748 1/20 0.37
GRIK1 P39086 1/20 0.35
EPHX2 P34913 1/20 0.35
PTPN5 P54829 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4969176 0.76 KMT2A (0.39) ALDH1A1MEN1KMT2AGPR35TMPRSS4
SCHEMBL29316655 0.74 CES2 (0.42) ALDH1A1MEN1KMT2ATMPRSS4MAPT
SCHEMBL7520231 0.73 ALDH1A1 (0.70) ALDH1A1MEN1KMT2AGPR35CA12
SCHEMBL391593 0.71 CES2 (0.45) ALDH1A1GPR35CA1CA2CES2
SCHEMBL194876 0.70 MEN1 (0.62) ALDH1A1MEN1KMT2AGRIK1
Hydrochloric Acid SCHEMBL9004750 0.69 MEN1 (0.60) ALDH1A1MEN1KMT2AGRIK1
SCHEMBL5118478 0.69 ALDH1A1 (0.68) ALDH1A1MEN1KMT2ACA12CA1
SCHEMBL14880120 0.68 CES2 (0.50) ALDH1A1KMT2ACES2
SCHEMBL4971330 0.66 PTPN5 (0.41) ALDH1A1MEN1KMT2ACA12CA1
SCHEMBL7524681 0.66 EPHX2 (0.78) ALDH1A1MEN1KMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed