SCHEMBL29330191

SCHEMBL29330191

COc1nc2c(c(Sc3ccc(F)cc3C(F)(F)F)n1)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 5/20 0.43
PARP1 P09874 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
HPGDS O60760 1/20 0.38
P2RX3 P56373 2/20 0.37
TGM2 P21980 1/20 0.37
ESR2 Q92731 1/20 0.37
MAPT P10636 2/20 0.37
PTPN11 Q06124 1/20 0.37
F12 P00748 1/20 0.36
RAF1 P04049 1/20 0.36
BRAF P15056 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NR1H2 P55055 1/20 0.36
RBP4 P02753 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29329976 0.90 PARP1 (0.42) MKNK1PARP1TNKS2PARP2HPGDS
SCHEMBL29330066 0.88 PARP1 (0.39) MKNK1PARP1TNKS2PARP2HPGDS
SCHEMBL30603339 0.86 MKNK1 (0.47) MKNK1PARP1TNKS2PARP2HPGDS
SCHEMBL29329977 0.82 P2RX3 (0.45) MKNK1P2RX3MAPT
SCHEMBL29330133 0.82 PTPN11 (0.35) MKNK1PTPN11RBP4
SCHEMBL21807309 0.78 PARP1 (0.43) MKNK1PARP1TNKS2PARP2P2RX3
SCHEMBL30603337 0.76 GPR119 (0.41) MKNK1PARP1TNKS2PARP2
SCHEMBL30603333 0.76 GPR119 (0.41) MKNK1PARP1TNKS2PARP2
SCHEMBL29330189 0.75 PARP1 (0.46) MKNK1PARP1TNKS2PARP2P2RX3
SCHEMBL29330192 0.75 PTPN11 (0.38) PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4400500-A1 HALOGEN-SUBSTITUTED PYRIDAZINONE COMPOUND AND APPLICATION THEREOF Medshine Discovery Inc. (CN) 2024-07-17 EP disclosed