SCHEMBL29329976

SCHEMBL29329976

CC(C)(C)OC(=O)N1CCc2c(nc(Cl)nc2Sc2ccc(F)cc2C(F)(F)F)C1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
MKNK1 Q9BUB5 5/20 0.41
ESR2 Q92731 1/20 0.39
TRPC5 Q9UL62 3/20 0.38
HPGDS O60760 1/20 0.38
RORC P51449 1/20 0.37
TGM2 P21980 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
PTPN11 Q06124 1/20 0.37
P2RX7 Q99572 1/20 0.37
F12 P00748 1/20 0.36
RAF1 P04049 1/20 0.36
BRAF P15056 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29330191 0.90 MKNK1 (0.43) PARP1TNKS2PARP2MKNK1ESR2
SCHEMBL29330066 0.86 PARP1 (0.39) PARP1TNKS2PARP2MKNK1ESR2
SCHEMBL30603339 0.86 MKNK1 (0.47) PARP1TNKS2PARP2MKNK1TRPC5
SCHEMBL21807357 0.83 TRPC5 (0.51) PARP1TNKS2PARP2MKNK1ESR2
SCHEMBL29329977 0.79 P2RX3 (0.45) MKNK1
SCHEMBL29330275 0.78 MKNK1 (0.48) MKNK1ESR2TRPC5HPGDSP2RX7
SCHEMBL21807251 0.76 TRPC5 (0.44) PARP1TNKS2PARP2ESR2TRPC5
SCHEMBL21807166 0.76 TRPC5 (0.43) PARP1TNKS2PARP2MKNK1ESR2
SCHEMBL30603333 0.76 GPR119 (0.41) PARP1TNKS2PARP2MKNK1GPR119
SCHEMBL30603337 0.76 GPR119 (0.41) PARP1TNKS2PARP2MKNK1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4400500-A1 HALOGEN-SUBSTITUTED PYRIDAZINONE COMPOUND AND APPLICATION THEREOF Medshine Discovery Inc. (CN) 2024-07-17 EP disclosed