SCHEMBL2933638

SCHEMBL2933638

COc1cccc(-c2c(C)cccc2C(=O)N2C[C@H]3C[C@H]3[C@H]2C(N)=O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.39
HPGD P15428 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
PARP1 P09874 1/20 0.36
PAX8 Q06710 2/20 0.36
KLK3 P07288 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
SLC9A1 P19634 1/20 0.36
PDE4B Q07343 1/20 0.36
MAOB P27338 1/20 0.35
CPS1 P31327 1/20 0.35
IKBKB O14920 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
DHODH Q02127 1/20 0.35
SCD5 Q86SK9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2925421 0.88 CFD (0.43) HCRTR1HCRTR2DHODH
SCHEMBL2929167 0.88 KDM4E (0.41) NPC1HPGDRAB9ASMN1; SMN2KDM4E
SCHEMBL2933639 0.86 PAX8 (0.39) NPC1HPGDRAB9ASMN1; SMN2KDM4E
SCHEMBL2924242 0.86 FABP4 (0.42) HPGDKDM4EALDH1A1HCRTR1HCRTR2
SCHEMBL2931039 0.85 HCRTR2 (0.39) PDE4BHCRTR1HCRTR2
SCHEMBL2930073 0.85 PDE4B (0.37) SLC9A1PDE4BHCRTR1HCRTR2
SCHEMBL2931529 0.85 HCRTR1 (0.46) NPC1HPGDRAB9ASMN1; SMN2KDM4E
SCHEMBL2931138 0.85 HCRTR1 (0.40) NPC1HPGDRAB9ASMN1; SMN2KDM4E
SCHEMBL2923504 0.83 PAX8 (0.38) PAX8TRPV1IKBKBHCRTR1HCRTR2
SCHEMBL2925366 0.83 HCRTR1 (0.39) PARP1TRPV1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed