SCHEMBL2933639

SCHEMBL2933639

COc1cccc(-c2c(C)cccc2C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 2/20 0.39
TRPV1 Q8NER1 1/20 0.37
BRD4 O60885 1/20 0.36
ABL1 P00519 1/20 0.35
EGFR P00533 1/20 0.35
SRC P12931 1/20 0.35
ABL2 P42684 1/20 0.35
NPC1 O15118 3/20 0.35
MAPT P10636 2/20 0.35
RAB9A P51151 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GRIN2B Q13224 3/20 0.35
THRB P10828 1/20 0.35
PRCP P42785 1/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2925423 0.89 CFD (0.40)
SCHEMBL2929170 0.87 KDM4E (0.43) PAX8TRPV1ABL1EGFRSRC
SCHEMBL2924244 0.87 CYP46A1 (0.39) PRCPHTR2B
SCHEMBL2931040 0.86 HCRTR2 (0.40)
SCHEMBL2930074 0.86 SLC6A7 (0.35)
SCHEMBL2933638 0.86 NPC1 (0.39) PAX8TRPV1BRD4NPC1MAPT
SCHEMBL2931139 0.85 HCRTR1 (0.39) PAX8TRPV1ABL1EGFRSRC
SCHEMBL2931530 0.85 HCRTR1 (0.46) PAX8ABL1EGFRSRCABL2
SCHEMBL2923507 0.83 PAX8 (0.39) PAX8TRPV1GRIN2B
SCHEMBL2925368 0.83 HCRTR1 (0.41) TRPV1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed