SCHEMBL29344739

SCHEMBL29344739

COc1ccc(CN(C)c2cc(Nc3cc(F)cc4c3OCCO4)nc3c(C(C)C)cnn23)cc1OC

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 11/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
CDK2 P24941 4/20 0.32
CDK9 P50750 1/20 0.32
ALDH1A1 P00352 2/20 0.32
P2RX7 Q99572 1/20 0.32
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CCNE1 P24864 1/20 0.31
HIF1A Q16665 1/20 0.31
EPAS1 Q99814 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29344741 0.94 CXCR3 (0.32) CXCR3GPBAR1ALDH1A1P2RX7LMNA
SCHEMBL29344736 0.93 CXCR3 (0.32) CXCR3GPBAR1ALDH1A1P2RX7LMNA
SCHEMBL29344747 0.92 P2RX7 (0.30) CDK2P2RX7
SCHEMBL29344717 0.91 CDK2 (0.33) CDK2CDK9CCNE1
SCHEMBL29344871 0.90 PTPN1 (0.34) CXCR3GPBAR1ALDH1A1P2RX7LMNA
SCHEMBL29344744 0.85
SCHEMBL29344684 0.84 POLB (0.30)
SCHEMBL29344732 0.81 P2RX7 (0.31) P2RX7
SCHEMBL23351255 0.81 ALDH1A1 (0.32) ALDH1A1P2RX7
SCHEMBL29344724 0.81 ALDH1A1 (0.31) ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024151992-A1 PREPARATION OF A TYK2 INHIBITOR VENTYX BIOSCIENCES, INC. (US) 2024-07-18 WO disclosed