SCHEMBL29356372

SCHEMBL29356372

NS(=O)(=O)c1ccccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 9/20 0.56
CA1 P00915 7/20 0.56
CA9 Q16790 7/20 0.56
CA6 P23280 5/20 0.56
CA7 P43166 5/20 0.56
CA5A P35218 5/20 0.56
CA12 O43570 5/20 0.56
CA4 P22748 4/20 0.56
CA5B Q9Y2D0 4/20 0.56
CA14 Q9ULX7 3/20 0.56
CYP2C9 P11712 1/20 0.56
PTGES2 Q9H7Z7 6/20 0.53
GAA P10253 1/20 0.48
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
LMNA P02545 1/20 0.47
HSD11B1 P28845 1/20 0.46
CA3 P07451 2/20 0.45
MAOB P27338 1/20 0.45
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL121865 1.00 CA2 (0.56) CA2CA1CA9CA6CA7
Hydrochloric Acid SCHEMBL27864427 0.98 CA2 (0.54) CA2CA1CA9CA6CA7
SCHEMBL2323386 0.98 CA2 (0.54) CA2CA1CA9CA6CA7
SCHEMBL2323381 0.98 CA2 (0.54) CA2CA1CA9CA6CA7
SCHEMBL29578190 0.81 PTGES2 (0.64) CA2CA1CA9CA6CA7
SCHEMBL742940 0.81 PTGES2 (0.64) CA2CA1CA9CA6CA7
SCHEMBL11647231 0.81 CA1 (0.52) CA2CA1CA9CA6CA7
SCHEMBL202947 0.81 CA2 (0.70) CA2CA1CA9CA6CA7
SCHEMBL28407818 0.81 CA2 (0.47) CA2CA1CA9CA6CA7
SCHEMBL30697126 0.79 HSD11B1 (0.59) GAATSHRHSD17B10LMNAHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078091-A1 Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer AMGEN INC (US) 2026-03-19 US disclosed
EP-4661966-A1 COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF Type6 Therapeutics, Inc. (US) 2025-12-17 EP disclosed
US-12479818-B2 Treatment of fibrosis with IRE1 small molecule inhibitors CORNELL UNIVERSITY (US) 2025-11-25 US disclosed
EP-3707126-B1 IRE1 SMALL MOLECULE INHIBITORS UNIV CORNELL (US) 2025-05-14 EP disclosed
US-20240425477-A1 IRE1 SMALL MOLECULE INHIBITORS CORNELL UNIVERSITY 2024-12-26 US disclosed
EP-4469442-A1 1,2,3-TRIAZOLE CARBONYL SULFONYLAMIDE COMPOUNDS AND USE THEREOF PI Industries Ltd. (IN) 2024-12-04 EP disclosed
US-20240300892-A1 Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer AMGEN INC (US) 2024-09-12 US disclosed
US-12071424-B2 IRE1 small molecule inhibitors CORNELL UNIVERSITY (US) 2024-08-27 US disclosed
WO-2024167848-A1 COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF TYPE6 THERAPEUTICS, INC. (US) 2024-08-15 WO disclosed
US-11945784-B2 IRE1 small molecule inhibitors CORNELL UNIVERSITY (US) 2024-04-02 US disclosed
CN-116981663-A Modulators of FPR1 and methods of use thereof 百放开曼有限公司 2023-10-31 CN disclosed
US-20230271935-A1 IRE1 SMALL MOLECULE INHIBITORS CORNELL UNIVERSITY 2023-08-31 US disclosed
WO-2023144711-A1 1,2,3-TRIAZOLE CARBONYL SULFONYLAMIDE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2023-08-03 WO disclosed
US-11634403-B2 IRE1 small molecule inhibitors CORNELL UNIVERSITY (US) 2023-04-25 US disclosed
CN-112694473-B 7, 9-disubstituted berberine structural analogue and preparation method and application thereof 南京林业大学 2022-09-20 CN disclosed
US-20220251065-A1 IRE1 SMALL MOLECULE INHIBITORS CORNELL UNIVERSITY 2022-08-11 US disclosed
US-20220227730-A1 TREATMENT OF FIBROSIS WITH IRE1 SMALL MOLECULE INHIBITORS CORNELL UNIVERSITY 2022-07-21 US disclosed
US-20220169611-A1 Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer AMGEN INC (US) 2022-06-02 US disclosed
US-20220024878-A1 IRE1 SMALL MOLECULE INHIBITORS CORNELL UNIVERSITY 2022-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230271935-A1 IRE1 SMALL MOLECULE INHIBITORS XBP1, ERN2, ERN1 CA2 4217/4885CA1 4652/4885CA9 4397/4885
US-20240300892-A1 Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer MDM2, TP53, CDKN1A CA2 3641/4885CA1 3382/4885CA9 3326/4885
US-20240425477-A1 IRE1 SMALL MOLECULE INHIBITORS XBP1, ERN2, ERN1 CA2 4217/4885CA1 4652/4885CA9 4397/4885
US-20260078091-A1 Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer TP53, HIF1AN, MDM2 CA2 535/4885CA1 1069/4885CA9 1154/4885
US-11634403-B2 IRE1 small molecule inhibitors XBP1, ERN2, ERN1 CA2 4217/4885CA1 4652/4885CA9 4397/4885
US-20220169611-A1 Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer MDM2, TP53, CDKN1A CA2 3641/4885CA1 3382/4885CA9 3326/4885
US-20220227730-A1 TREATMENT OF FIBROSIS WITH IRE1 SMALL MOLECULE INHIBITORS XBP1, DDIT3, ATF4 CA2 4160/4885CA1 4828/4885CA9 4598/4885
US-11945784-B2 IRE1 small molecule inhibitors XBP1, ERN2, ERN1 CA2 4217/4885CA1 4652/4885CA9 4397/4885
US-12071424-B2 IRE1 small molecule inhibitors XBP1, ERN2, ERN1 CA2 4217/4885CA1 4652/4885CA9 4397/4885
US-20220251065-A1 IRE1 SMALL MOLECULE INHIBITORS XBP1, ERN2, ERN1 CA2 4217/4885CA1 4652/4885CA9 4397/4885
US-12479818-B2 Treatment of fibrosis with IRE1 small molecule inhibitors XBP1, DDIT3, HSP90B1 CA2 4134/4885CA1 4827/4885CA9 4583/4885
US-20220024878-A1 IRE1 SMALL MOLECULE INHIBITORS XBP1, ERN2, ERN1 CA2 4217/4885CA1 4652/4885CA9 4397/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.